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"Luminal": ntuziaka maka ojiji nke nwa ọhụrụ

Gịnị bụ ọgwụ "Luminal"? Ntuziaka na-egosi nke a ọgwụ ga-atụle n'okpuru. Anyị na-akọwa na pharmacological Njirimara nke ọgwụ, ya mmetụta na contraindications.

The mejupụtara nke ọgwụ na ụdị

Na e dere a ọgwụ ọjọọ, "Luminal"? Ntuziaka maka ojiji na-akọ na na mejupụtara nke a Nwa-agụnye nọ n'ọrụ mgwa dị ka phenobarbital. -Atụle n'aka na-agụnye ndị na-esonụ ọzọ mmiri: nduku starch, gelatin, talc na calcium stearate.

Nkwadebe "Luminal", na-egosi nke a na-ọkọnọ dịrị gaba n'ime ebe, a na-ahịa na ụdị a powder zubere maka ihe ngwọta maka ogwu ogbugba. Ọzọkwa ngwá ọrụ a nwere ike zụrụ n'ụdị mbadamba 100 mg, nke na-juru n'ọnụ na cell ngwe na nkwakọ mere akwụkwọ, karị.

The ọgwụgwọ mmetụta nke ọgwụ

Gịnị bụ nke a na nkà mmụta ọgwụ dị ka "Luminal"? Ntuziaka maka ojiji rụrụ ụka na a usọbọ nwere ogwuura, hypnotic na anticonvulsant mmetụta.

E lee ya anya agwọ ọrịa ike nke na-agbalịsi suppressive edinam (na-abụghị nhọrọ) na mmadụ ụjọ usoro, na-inhibit ụfọdụ ebe (na-emekarị sensory) cortex belata locomotor ọrụ, ịzụlite iro ụra na ogwuura.

Drug "Luminal" ntụziaka na ngwa nke nke bụ na akwụkwọ tojupụtara bụ a nnọọ ike barbiturate. Ya ogwuura-hypnotic Njirimara bụ n'ihi mgbochi nke ọrụ nke mkpụrụ ndụ, nke rụọ ọrụ ndị reticular guzobere nke nuclei nke thalamus, brainstem, si otú inhibit na mmekọrịta nke kwuru owuwu na-arịa ọrịa cortex.

atụmatụ ọgwụ

Gịnị dị ịrịba ama iji ọgwụ "Luminal"? Ntuziaka maka ojiji (mụrụ ọhụrụ bụ ụzọ kenyere ukwuu mgbe) na-ekwu na ụra kpatara nke a barbiturate, jiri ya tụnyere saline nwere a kpamkpam dị iche iche Ọdịdị. Dị ka a na-achị, na mmepe nke hypnotic mmetụta na etinye a ọgwụ maka 35-65 nkeji na dịruru maka 6-9 awa.

Anyị nwere ike ikwu na usọbọ n'okpuru echiche ngosi akpọ anticonvulsant Njirimara. Ha na-mere site mmetụta nke ọgwụ na ụfọdụ ebe nke ụjọ usoro. Mgbe na-eji nke a ọgwụ na ọrịa ebelata neuronal excitability na epileptogenic mpaghara nke na-egbochi ntoputa na mgbasa nke pulses. Ọzọkwa na ndabere nke "Luminal" na-ekwu igbochi elu ugboro discharges akwara ozi, na-abawanye na nbata-uzọ nke eletriki mmalite na moto region nke ụbụrụ cortex.

Ke adianade do, maka nyere ọgwụ e ji a obere analgesic mmetụta na antigiperbilirubinemichesky. Ọzọkwa bụghị chịrị si ike nke ahụ Jeremaya mere ka na-egbu mgbu stimuli.

Obere Dosages "luminal" nwere a calming mmetụta, na elu na--ugnetayut ume medulla emmepe na t. D.

kinetic atụmatụ

ma ọgwụ na-etinye obi gị dum, "Luminal"? Ntuziaka maka ojiji na-akọ na n'ime ahụ ya dabara a na-adịghị na ha zuru ezu absorption. The bioavailability nke gị n'ụlọnga bụ banyere 80%, na nkekọ na-plasma-edozi - banyere 30%.

The n'ọrụ mgwa nke ọgwụ penetrates na mmiri ara nne, nakwa dị ka Plasenta. Ọzọkwa, ọ nwere ike na-ekesa na nwa ebu n'afọ na arọ.

Excretion "luminal" pụtara via akụrụ na-agbanweghi agbanwe ụdị ma ọ bụ n'ụdị metabolites. N'ihi phenobarbital ji nnọọ nnọọ ìgwè. Ọrịa nke akụrụ na-akpata prolongation nke edinam.

Drug "Luminal": egosi maka ojiji

Weere a ọgwụ na-kenyere ọ bụghị naanị ndị okenye, ma ụmụaka na mụrụ ọhụrụ. Dị ka a na-achị, ọ na-eji maka:

  • hyperbilirubinemia;
  • akwụkwụ na-adọ;
  • tetanus (maka adjuvant ọgwụ);
  • ọgwụgwọ nke nnukwu convulsive ọdịdọ.

Anyị apụghị ikwu na ngwá ọrụ a nwere ike kenyere ngụkọta ọgwụgwọ dị ka a ogwuura ọgwụ iji kpochapụ nchegbu, egwu na nrụgide.

Bans ojiji

Ugbu a ị maara n'okpuru ihe ọnọdụ ọrịa na-kenyere a na nkà mmụta ọgwụ "Luminal". Egosi maka ojiji nke a ọgwụ e depụtara n'elu. Banyere contraindications, mgbe ahụ, ha na-ebu dị ka:

  • elu uche ọgwụ;
  • oké umeji akụrụ mmebi;
  • dị iche iche nke porphyria;
  • lactation na ime.

Agwọ ọrịa "Luminal": ntuziaka maka ojiji maka ụmụaka na ndị okenye

The ojiji nke a ọgwụ ga-nditịm gosiri. Ya iji na-achọ nhọrọ nke ahaziri ọgwụgwọ Usoro, onunu ogwu, na oge nke nke na-adabere ọ bụghị nanị na ụdị eruba nke ọrịa, ma na ọrịa afọ na ndị ọzọ e ji mara.

Dị ka ntụziaka, nkezi otu dose akuko ngwaọrụ n'ihi na ndị okenye bụ 10-200 mg. Were dị otú ahụ ọgwụ kwesịrị 1-3 ugboro n'ụbọchị.

Ma nwa ọhụrụ ụmụ, ha ọgwụ dose a gbakọọ dabeere na ahu arọ (1-10 mg / n'arọ ahu arọ ugboro atọ n'ụbọchị).

Ọ bụrụ na-na-emeso ọrịa n'ụdị nke ọgwụ infusion, na onunu ogwu maka okenye bụ 100-1400 mg (igba ogwu n'akwara infusion), ma ọ bụ 10-200 mg (n'ihi na intramuscular injection).

Ngụkọta oge nke dose of isiokwu nke ụmụ ọgwụ a na-rụrụ dabeere na ịdị arọ nwatakịrị.

Dị ka ndị ọkachamara, mgbe igba ogwu n'akwara ochichi, "luminal" ya kacha mmetụta ruru n'ime 35 nkeji.

mmetụta

Ime ọjọọ na ahụ mmadụ ọgwụ "Luminal"? Ntuziaka maka ojiji (site na-asọ ya pụtara bụghị gosiri) rụrụ ụka na ọgwụgwọ nke data ọgwụ ọrịa nwere ike ịzụlite a dịgasị iche iche nke mmetụta na-emetụta ihe nile dị oké mkpa akụkụ na usoro. Oghom mgbaàmà adịghị ike, ike ọgwụgwụ, na-ehi ụra, ịda mbà n'obi na ataxia. Ọ dịkwa ike mmepe nke thrombocytopenia, agranulocytosis, nfụkasị Jeremaya na-anaghị ekwe nke calcium metabolism.

ikpe nke ovadozu

Na ihe ovadozu nke "TMB" ọrịa nke ukwuu mgbe nwere isi ọwụwa, nystagmus, dizziness, ataxia, nsogbu iku ume, lethargy, adịghị ike, okwu impairment, iro ụra, mgbanwe ahu okpomọkụ, agụụ, ọbara mgbali na ndị ọzọ na ọdịda. Na ihe mgbagwoju ikpe, e nwere: bradycardia ma ọ bụ tachycardia, akpa ume edema, mgbagwoju anya, arrhythmias, Coma, oyi baa na na.

Iji kpochapụ ndị a mgbaàmà bụ ọgwụ gastric lavage nakwa dị ka detoxification ọgwụgwọ.

ọgwụ interactions

Ngwa nke na-ewere gị n'ụlọnga na Nchikota na ọgwụ ọjọọ mwute HC, methylphenidate ma ọ bụ Mao inhibitor enwekwu ịta nke ya nọ n'ọrụ mgwa na mejupụtara nke plasma, nke na-eduga na ụba na-egbu egbu mmetụta na mgbochi nke NA.

The Nchikota "Luminal" na corticosteroids, chloramphenicol, corticotropin, dacarbazine, cyclosporine, digitalis glycosides, quinidine, metronidazole, tricyclic antidepressants, carbamazepine, mgbochi ịnara ọkwá n'ike, nke succinimides otu, doxycycline, anticoagulants, chlorpromazine, fenoprofenom, vitamin D na phenylbutazone nwere ike belata oge edinam na ike nke ndị a ọgwụ ọjọọ eme ihe na-amụba ha metabolism, nakwa dị ka ibu arọ na imeju.

Concurrent ọgwụgwọ na acetazolamide nwere ike na-eme ka mmepe nke rickets na osteomalacia. Valproic acid enhances phenobarbital ịta na ọbara, nke na-akpata a akpọ ogwuura na lethargy.

Eji "luminal" ọnụ na nimodipine, "Verapamil" na felodipine ebelata ha ịta ke iyịp.

The Nchikota nke agwọ ọrịa na maprotiline enhances ya inhibitory utịp ke NA, ebelata mmetụta nke anticonvulsant barbiturates na convulsive mbata.

Active mgwa "luminal" paracetamol pụrụ ibelata arụmọrụ na-akwalite mmepe nke hepatotoxicity. Mgbe jikọtara folic acid na-ebelata arụmọrụ nke phenobarbital.

Pyridoxine lowers ọbara ịta nke phenobarbital, na primidone, felbamate na, ọzọ, welie ya.

Analogs nke ọgwụ na ya price

Ihe bụ isi ọgwụ na-atụle analogues dị otú ahụ dị ka "Barbinal" na "Dormiral".

Cost mbadamba "Luminal" (100 mg, 10 PC.) Of 1100 rubles na n'elu.

kpọmkwem ozi

Imekotaotuugbo n'ikuku "luminal" si ethanol na ethanol-n'aka ike budata welie inhibitory mmetụta nke ọgwụ na ụjọ usoro nke ọrịa. Ya mere, na-aba ọṅụṅụ na ndị ọzọ ọgwụ tinctures na mmanya n'oge ọgwụgwọ ndị a elekọta mmadụ na-contraindicated.

Nyocha

Kasị reviews nke a nkwadebe ahapụ nne na nna nke ụmụaka. Ha na-ekwu na ọgwụ "Luminal" ezi agha na ọrịa ndị dị ka Akwụkwụ na-adọ na convulsive ọnọdụ. Ọ na-abụkarị ndị ọgwụ na-eji dị ka akụkụ nke Nchikota ọgwụ, zuo ezu ya ahụ mgbu.

Ọtụtụ ọrịa na-ekwu na elu arụmọrụ nke ọgwụ "Luminal". Otú ọ dị, ozugbo ahụ ha kwuru na n'elu nnata nke ego ga-erube nnọọ na-eso usoro onunu ogwu na ya Nchikota na ndị ọzọ ọgwụ ọjọọ.

Mgbe ụfọdụ, na-ewere a na nkà mmụta ọgwụ na-eji maka ọgwụgwọ nke ndị na-vaskụla dystonia, nke na-esonyere oké nke egwu ọgụ. Ọgwụgwọ nke ngwá ọrụ a na-enyere aka normalize ọnọdụ nke onye ọrịa, karịsịa ma ọ bụrụ na ọ bụ ihe ọzọ ọgwụ, dilates ọbara arịa na aka apịajighị apịaji.

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