Ahụ ike, Preparations
"Olanzapine": analogues, ọgwụ nkọwa, ntuziaka maka ojiji
Maka ọgwụgwọ nke isi mgbaka na imetụ mmadụ n'isi eji ọgwụ ọjọọ eme ihe na-adabere umi olanzapine. E nwere ọtụtụ ọgwụ ọjọọ dị iche iche na ahia aha, ma otu antipsychotic mmetụta. One dị otú ahụ ọgwụ ọjọọ bụ ọgwụ "olanzapine" analogs nwere ya mejupụtara ngụkọta n'ọrụ mgwa.
Description of nkwadebe
Nke a na-eme site na antipsychotic gị n'ụlọnga "ALSI Pharma" ZAO ka a ìhè edo edo mbadamba, na udi nke yiri a cylinder biconvex.
Ọdịdị nke ọgwụ na-etolite na-adịghị ejekwa Efrata, nke na-agụnye microcrystalline cellulose ụdị, lactose monohydrate, krospovidonovy dịanyā, magnesium stearate. Ha nọmba enwekwu na abụọ, atọ ma ọ bụ ugboro anọ, dabere na onunu ogwu olanzapinovoy.
The mbadamba na-juru n'ọnụ niile doses nke 7 iberibe na blisters na a mkpọ nke nwere ike ịbụ 4 ma ọ bụ 8 iberibe.
Pụtara "olanzapine" User Ngwa akọ na antipsychotic neuroleptic ọgwụ ọjọọ nke igosipụta mmekọrita maka serotonin, dopamine, muscarinic, adrenergic na histamine ihe nnabata guzobere.
Bibiri belata excitatory ọrụ nke mesolimbic dopaminergic akwara ozi, nwere obere ọrụ striatal akwara conduction, nke achịkwakwa ọrụ engine. Mgbada n'usoro ike ot echebe-aghọ nkọ, ma ọ bụrụ na ị na-eji a ala onunu ogwu enweghị na-eme cataleptic ụra.
Medicine "Olanzapine" enwekwu anxiolytic nrụpụta nke ule ọrụ "anxiolytic" ka a nọ na-agba ọsọ. Eburu ịkwụsị ịṅụ na-adịghị mma na-arụpụta ka delusions na hallucinatory ọhụụ.
Gịnị na-eji
Mbadamba "olanzapine" mmetụta dọgburu on schizophrenic ala na-etoru ogo mmadụ na nnukwu ogbo, dị ka a njigide na ruo ogologo oge protivopovtornogo ọgwụgwọ. Ha na-eji psychotic aghara na a na-amị mkpụrụ ihe ịrịba ama nke delusions, hallucinatory ọhụụ na-adịghị mma mgbaàmà ndị dị otú ahụ dị ka obi abadaba, na-ebelata mmadụ ịrịba omume, depletion nke olu ngwa.
Drug tutu amama nlọghachite nke ọdịdọ na imetụ mmadụ n'isi, ma ọ bụrụ na mbadamba nkume ọma na-emeso manic nkebi.
Nkwadebe "olanzapine" nyere ndị okenye na bipolar affective ọrịa n'ụdị monotherapy ma ọ bụ na njikọ na ọgwụgwọ nwere lithium ion ma ọ bụ valproic acid. The ọgwụ na-eji na-emeso nnukwu manic ma ọ bụ mbuaha iche nke omume ahụ nwere ike ime psychotic atụmatụ, dị ka nke ọma dị ka nwere a ngwa ngwa mgbanwe nkebi.
Pụtara jikọtara na fluoxetine ọgwụ maka dara ya mbà ọnọdụ na-metụtara imetụ mmadụ n'isi.
Usoro ojiji
Medicine "olanzapine" User ngwa na-atụ aro na ụbọchị site na 0,005 na 0,02 g ọnụ enweghị n'ịnọgide ike mode.
schizophrenic ala Okenye ọrịa emeso ya na mbụ kwa onunu ogwu nke 0,010 g
Adult nnukwu Mania, imetụ mmadụ n'isi ji, wepụrụ kwa ego nke olanzapine na 0.015 g, nke a na-ndinọ ozugbo. Ọ bụrụ na mbadamba nkume na-eji njigide metụtara njikọ na ọgwụ dabeere na lithium ion ma ọ bụ valproic acid, mgbe ndinọ na a kwa ụbọchị dose nke 0,010 g kwa mgbe.
Dara ya mbà Filiks ke ịghọ okenye ruru imetụ mmadụ n'isi, dochie kwa ego nke 0,005 g, na-achọkwa na 0,020 g fluoksetinovogo umi. Ọ bụrụ na e nwere mkpa, mgbe ahụ, kwe ukpụhọde nke dosing nke ọgwụ.
Agadi ọrịa na-ekwe omume nke ukwu ihe iyi egwu gbasara akụrụ insufficiency ma ọ bụ na-adịghị ala ala imeju dị ka mgbe e nwere ihe ize ndụ ndị a na-nwaanyị okike, senail ebighi-mgbe deceleration mgbanwe olanzapine ya mbụ kwa ụbọchị ego na-ebelata ka 0,005 g
a ngwaọrụ
Agwọ ọrịa "Olanzapine" ogbo nwere dị iche iche ahia aha. Ha na-emepụta site ma anụ ụlọ na ndị mba ọzọ na-emepụta.
N'etiti Russian Nsukka nke atụ ogho-apụ ụlọ ọrụ 'ọgwụ ọjọọ Technologies "na ọgwụ" Olanzapine-TL ", na mbadamba ụdị 0,0025 g film ntekwasa.
Ọzọ anụ ụlọ ọgwụ bụ ụzọ nke "Olanzapine", arụpụtara site JSC "North Star". E nwere a mbadamba na a film mkpuchi na a dose nke 0,005 g
Russian factory "Kanonfarma Production" JSC emepụta ọgwụ "Canon nke olanzapine."
Israel na nkà mmụta ọgwụ bụ na nkà mmụta ọgwụ "Olanzapine Teva," emeputa ụlọ ọrụ "Teva Pharmaceutical Enterprise Co., Ltd.".
Slovenian analogue bụ pụtara "Zalasta Cu tab", na mbadamba nkume nke 0,015 g kara aka maka resorption. Mere site enterprise "Krka, Novo Mesto." Ọzọkwa data mepụtara ọgwụ "Zalasta" mbadamba.
Swiss ọgwụ analogue na-atụle "Zyprexa" dị ka a lyophilisate na vials, site na nke njikere ngwọta maka intramuscular ochichi, a dose of 0,010 na dispersible mbadamba ụdị 0.005 grams dị ọgwụ "Zyprexa Zidis". Ha na-emepụta site na "Eli Lilly Vostok SA". Na-emepụta ọgwụ ahịa e nwere "Zyprexa Adair" powdered agwọ ọrịa a na-akụzi 0,21 g
Polish ụlọ ọrụ nke "Polpharma" arụpụtara na nkà mmụta ọgwụ "Normiton" mbadamba na a n'ọbọ mkpuchi nke 0.005 g
Drug "Olanzapine" Hungarian ogbo mepụtara "Gedeon Richter" na-akpọ mbadamba "Parnasan" na-emepụta ọgwụ osisi "EGIS" mepụtara ọgwụ "Egolanza".
Description "Zalasta" ọgwụ
Nke a na-ezo aka antipsychotic neuroleptic. Ìhè odo mbadamba dị gburugburu, ubé biconvex udi na ọchịchịrị patches. E nwere ihe isii Dosages: 0,0025 g, 0,005 g, 0.01 g, 0,015 g na 0,02 g nke olanzapine. Ọzọ mmiri na-atụle na-adịghị ejekwa Cellactose, starch pregelatinized na ọka ụdị, dehydrated aerosilovy mgwa, magnesium stearate.
Akara mbadamba ụdị "Zalasta" ntụziaka ntuziaka na-akọwa notation n'ụdị a tụrụ atụ na-egosi nke usoro onunu ogwu. Consumer nchịkọta bụ contoured efere 7 mbadamba. The mkpọ nwere ike ịnwe 4 ma ọ bụ nke 8 nke ndị dị otú ahụ blisters.
Nke a neuroleptic gị n'ụlọnga na-egosipụta sara mbara pharmacological-eme. Antipsychotic mmetụta jikọtara interlock formations dopamine ihe nnabata ụdị. Ogwuura ọrụ mere site braking adrenoceptor saịtị na mejupụtara ndị reticular guzobere na mkpụrụ ndụ nke ụbụrụ azuokokoosisi.
Antiemetic ọrụ bụ na o kwere omume na-akwụsị D 2 ihe nnabata -dopaminovogo òkè na triga-ụdị mpaghara bụ nke dị na emetic center.
Hypothermic ọrụ a rụrụ site igbochi dopamine ihe nnabata formations nke umu ke hypothalamus.
Medicine "Zalasta" ntụziaka ntuziaka na-atụ aro iji na schizophrenic n'obiọma. Mbadamba na-enwe ike ifịk ifịk na-mgbanwe nke-adakarị mgbaàmà n'oge ogologo oge ọgwụgwọ nke ọrịa na mbụ mmetụta dị mma na ọgwụ.
Pụtara kpochapụ episodic Mania n'etiti ma ọ bụ mgbagwoju ụdị. Mbadamba omume aka ná ntị mkpachapụ ugboro ugboro ibu na imetụ mmadụ n'isi na ndị mmadụ na manic ngosipụta.
The ọgwụ na-zubere maka onu ochichi otu ugboro n'ụbọchị. nri ahụ adịghị emetụta absorption usoro nke olanzapine, nke-enye gị ohere iji mbadamba n'oge ọ bụla. N'elu kagbuo nke ọgwụ ga-eji nwayọọ nwayọọ belata dose.
Maka ọgwụgwọ nke schizophrenic ọrịa na-eji na mbụ dosing nke 0,010 grams kwa ụbọchị.
Ji nke Mania amalite emeso kwa ụbọchị dose nke 0.015 g, nke a na-ndinọ n'otu ngwa ma ọ bụ 0,010 grams mgbe jikọtara ndị ọzọ neuroleptics.
Ikwughachi mgbochi nke ihe imetụ mmadụ n'isi na attenuation nzọụkwụ a rụrụ ke akpan ekesa agwọ ọrịa 0,010 grams kwa ụbọchị. Ọ bụrụ na ndị mmadụ na-na ngwá ọrụ na-agwa okwu episodic Mania, maka nketa nke ọgwụ iji otu dose. Ọ dị mkpa ka dịkwuo ego nke ọgwụ na ihe omume nke ọhụrụ ma ọ bụ grouped episodic dara ya mbà ngosipụta, nakwa dị ka ịgbakwunye na ọgwụgwọ nke na ọnọdụ disruptions.
The kwa ụbọchị dose nke agwọ ọrịa iji kpochapụ schizophrenic ọrịa, manic ngosipụta na bipolar ọrịa ịdọ aka ná ntị akuko iji si 0,005 na 0,020 g, uru nke na-adabere na-adakarị kwa nke onye ọrịa.
Agadi ala mbụ onunu ogwu nke ruo 0.005 g na-adịghị gwara Otú ọ dị, ndị dị otú ahụ na-eme ga-etinyere ọrịa si afọ 65, ma ọ bụrụ na e nwere ihe ize ndụ ihe.
Description "Olanzapine Canon" ọgwụ
A edinam nke neuroleptic antipsychotic agwọ ọrịa dị na mbadamba ụdị ntekwasa na a n'ọbọ. Udi nke mbadamba nkume mechie abụọ convex ebupụta odo, esịtidem ọdịnaya nke otu na agba.
Ọ dị ihe abụọ Dosages: na 0,005 g na 0.01 g nke olanzapine. The inyeaka Efrata gụnyere hydroxypropyl cellulose na ala nnọchi, calcium hydrogen phosphate, croscarmellose sodium, mannitol, magnesium stearate.
N'ọbọ odo Opadry film a kpụrụ nke abụọ ụdị, polyvinyl mmanya, macrogol, talc, titanium dioxide, ígwè oxide.
Drug ọgwụgwọ kenyere impairments, maka inwe na itinye ogologo antirelapse okenye ọrịa na-ata ahụhụ site na schizophrenic ọrịa.
The na-agwọ na-rụrụ monotherapy na Nchikota itinye n'ọnọdụ na lithium compound na a siri ike n'ụdị manic ma ọ bụ mbuaha ji nke bipolar affective aghara, nke bụ okwu na psychotic na na ngwa ngwa na-agbanwe agbanwe n'ụzọ. Ọgwụ iji gbochie repetitions na ndị mmadụ na-emetụ n'isi ọrịa, ma ọ bụrụ na ọgwụ aka ịnagide manic ogbo.
Na ọgwụgwọ nke okenye na ịda mbà n'obi mere site imetụ mmadụ n'isi, nakwa dị ka anụ dara ya mbà ogo ngwọta "Canon Olanzapine", a neuroleptic, Enwere ike ikpokọta ozi nwere fluoxetine.
Ọ na-e jikwa ọnụ, ọ bụghị ịgbaso ihe oriri. Guide na-atụ aro na ọgwụgwọ onunu ogwu nke agwọ ọrịa, nke bụ ụbọchị, ọnụ ọgụgụ nke 0,005-0,020 n'aka na-ahọrọ n'otu n'otu n'ihi na onye ọ bụla ndidi dabere na-adakarị ịrịba ama.
Schizophrenic ọrịa okenye ọrịa emeso mbụ kwa dosing ọgwụ na 0.010 g, nke a na-ndinọ ozugbo.
Ọnọdụ imetụ mmadụ n'isi nnukwu Mania kpochapụ kwa onunu ogwu nke ọgwụ ka 0,015 g ma ọ bụ 0,010 g nke olanzapine jikọtara na mmadụ nwere lithium ion ma ọ bụ valproic acid.
Eme ojiji nke ihe imetụ mmadụ n'isi n'oge mbụ kwa dosing a rụrụ na 0.010 ọrịa e rụrụ ma ọ bụrụ na n'ikuku nke a agwọ ọrịa maka nnukwu Mania, ọ ga-anọgide na-eji ego na otu ichekwa.
Dara ya mbà ọrịa metụtara na imetụ mmadụ n'isi okenye ọrịa emeso ya na a Nchikota 0,005 g na 0,020 g nke olanzapine fluoksetinovyh preparations nke na-ndinọ na mgbede.
Antidepressive mmetụta nke ọgwụ gosi na ego nke si 0,006 na 0,012 grams na nkezi kwa ụbọchị dosing na 0,0074 g dose fluoksetinovyh ọgwụ àmà site 0,025 na 0,030 g Ọ bụrụ na e bụ mkpa, ọ bụ omume na-agụgharị dosing nke ma ọgwụ ọjọọ.
Therapeutic anụ ụdị ịda mbà n'obi na-wepụrụ a Nchikota 0,005 g na 0,02 g nke olanzapine fluoksetinovyh n'aka nke a na-ndinọ ozugbo na mgbede.
Description "Zyprexa" ọgwụ
Nke a neuroleptic emepụta mbadamba ụdị ntekwasa na a n'ọbọ. E nwere ihe anọ onunu ogwu Nwa: 0,0025 na 0,005, 0,010 na 0,0075 maka x, y nke bụ ihe kwesịrị ekwesị notation n'elu «LILLY 4112», «LILLY 4115», «LILLY 4116», «LILLY 4117".
-Adịghị ejekwa ozi Efrata n'ụdị lactose, hydroxypropylcellulose, crospovidone, microcrystalline cellulose ụdị Ọdịdị a kpụrụ nke magnesium stearate ọgwụ.
The mbadamba na-packaged ke blisters nke 7 iberibe na a mkpọ nwere 4 ngwe nkwakọ.
E nwekwara a ifriizi-Fikiere ụdị, zubere maka imewe nke intramuscular ngwọta. Yellow mmiri mmiri onunu ogwu 0.01g packaged n'ime vials. -Adịghị ejekwa ozi mmiri na-atụle lactose monohydrate na tartaric acid.
The ọgwụ na-egosipụta antipsychotic mmetụta.
The n'ọrụ mgwa nke agwọ ọrịa na-akpa àgwà dị ka ligand nke ejikọ na serotonin, dopamine, m-choline, H1-histamine na alpha1-ihe nnabata adrenozavisimymi formations. Olanzapine nwere a nhọrọ utịp ke ala nke limbic usoro.
Drug "Zyprexa" ntụziaka na ngwa na-adụ ọdụ iji na ike nkebi nke schizophrenic na psychotic ọrịa na-ebu doro anya ihe ịrịba ama nke delusions, ịmụ anya arọ nrọ, echiche ọrịa, obi ọjọọ, na enyo àgwà ma ọ bụ a na-ezighị ezi ụdị na ụdị mmetụta uche na-elekọta mmadụ na mwepu, ọrịa nke olu ngwa. The na nkà mmụta ọgwụ na-owụt maka mwepụ nke abụọ affective mgbaàmà mere site schizophrenic ọrịa.
Tablet "Zyprexa" ntụziaka ntuziaka tụrụ aro na-aṅụ ọnụ, n'oge ọ bụla. Early ọgwụgwọ nke otu dose bụ 0,010 g mesịa, kwa ụbọchị onunu ogwu àmà site 0,005 na 0,020 g, nke a na ekekọtara na symptomatic picture.
Intramuscularly agbara ọgwụ, ma ọ bụrụ na mkpa kwụsị na excitation psychomotor agwa ndị mmadụ na isi mgbaka, bipolar affective ọrịa na mgbaka.
Tupu ojiji, lyophilisate e diluted na 2.1 ml injectable okenye ọkara. A doro anya ihe ngwọta na a odo tinge.
The ụjọ obi ụtọ nke schizophrenic na imetụ mmadụ n'isi gbapụ na a otu-dose of 0,010
Ịtụle ugbu a na ọgwụgwọ ọrịa, ugboro ugboro ochichi nke onunu ogwu 0,010 g rụrụ mgbe 120 min si akpa ngwa na ndị na-esonụ 0,010 g iwesa mgbe 240 nkeji nke abụọ ngwa.
N'ihi na n'ihu ọgwụgwọ ọgwụ ọjọọ, "Zyprexa" kwagara ya mbadamba ụdị na a onunu ogwu nke si 0,005 na 0,020 g
Oyobio na mgbaka ewepụ ke otu intramuscular dose of 0,0025 Ịtụle adakarị foto nke ọrịa, nke abụọ ochichi onunu ogwu 0.005g rụrụ mgbe 120 nkeji si akpa ngwa.
Product nkọwa "Adair Zyprexa"
E agwọ ọrịa "olanzapine" analogs na-emepụta na ntụ ntụ ụdị site 0,405 g nke olanzapine na vials na a mgbaze ntụtụ na agịga.
Pụtara "Adair Zyprexa" na-ezo aka antipsychotic neuroleptic ọgwụ ọjọọ ọrụ.
Ọgwụ suppresses arịa ọrịa, na-eji maka njigide na ogologo okwu ọgwụgwọ nke schizophrenic protivopovtornogo na uche mgbanwe na mgbaàmà nke elu-mkpụrụ na ụdị delusions, hallucinatory ọhụụ na-adịghị mma obi abadaba, depleted na olu ngwa.
Ọgwụ na-emeso oké manic na jikọtara ji nke ihe imetụ mmadụ n'isi, n'oge nke ọ bụ omume psychotic atụmatụ na a ngwa ngwa mgbanwe na nkebi.
Mbụ kwa onunu ogwu na-eji 0.010 ma ọ bụ 0.015, kwa ụbọchị ego nke ọgwụ ahọrọ maka onye ọ bụla ndidi n'otu n'otu, na-ewere n'ime akaụntụ na-adakarị picture. A na-eji ọgwụgwọ kwa ụbọchị dose nke si 0,005 na 0,020 g
Ịba na onunu ogwu bụ nanị kwe omume na-arụpụta nke nyocha. Amụba ego nke ọgwụ a rụrụ nkebi, ụbọchị ọ bụla.
Agadi ọrịa, na mbụ kwa ụbọchị dose na ọnụnọ nke ezughi oke akụrụ ọrụ na imeju na ikpo 0.005 g
eri analogues
Large agwaogwa nke antipsychotics enye gị ohere ịhọrọ nri ọgwụ, nke kwesịrị ekwesị dị na àgwà na-eri. Ọgwụ "Olanzapine" a dịtụ obere price. Packaging nke mbadamba nwere ike zụta maka 290 rubles.
Drug "Zalasta" price bụ site 1370 rubles.
Oké ọnụ ụzọ na-ewere ọgwụ "Zidis Zyprexa." Maka ngwaahịa ngwugwu mkpa iji kwụọ ụgwọ 2370 rubles. analọg uru nke "Ku-Tab Zalasta" bụ 1075 rubles.
On na nkà mmụta ọgwụ "Zyprexa" price natara ọjọọ reviews. A mkpọ 28 mbadamba efu 4760 rubles.
N'ihi na-enweghị ka ìgwè dị iche iche ga-abụ dị ọgwụ "Olanzapine", nke bụ akụkụ dị nta nke price.
Echiche nke ọrịa
About ọgwụ "Olanzapine" reviews nwere ike nụrụ ma nke oma ma na-ezighị ezi. Ọtụtụ ọgwụ na-enyere aka ịnagide ịda mbà n'obi na ibelata ego nke na-ezighị ezi echiche mgbe a ụbọchị ole na ole nke ọgwụgwọ. Ọ a na-ewere otu n'ime eme nke neuroleptics, nke calms ọrịa, eliminates egwu na nchegbu.
N'etiti ọghọm emit achọghị mmetụta nke na-metụtara a slowing nke metabolism, dapụtara na ụba ahu arọ nke onye ọrịa. Somnolence, asthenia syndrome, dizziness, orthostatic ọbara nwere ike idebe ụdị nsogbu ịzụlite adụ anụ ahụ ọzịza na nkụ nke mucous membranes.
N'ihi na ụfọdụ ndị ọrịa, ọbụna a obere dose nke nkà mmụta ọgwụ bụ a siri ike ogwuura, nke ha na-ehi ụra ruo 12 awa a ụbọchị.
Ahụ mmadụ dị iche iche, Otú ọ dị, na mbadamba-akpa àgwà dị iche iche nke ọ bụla ndidi. N'ihi na nhọrọ nke kwesịrị ekwesị ngwaọrụ mkpa ịkpọ onye dọkịta.
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