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Ọgwụ "Chlorpromazine": reviews nke dọkịta, ntuziaka maka ojiji, mejupụtara na nkọwa

Antipsychotic ọgwụ - a psychotropic ọgwụ ọjọọ, bụ ndị e mere maka ọgwụgwọ nke psychotic ọrịa. Ọ ga-kwuru na omenala aha nke ndị dị otú ahụ ọgwụ ọjọọ eme ihe - neuroleptics. Ndị a ọgwụ ọjọọ nwere ike n'ụzọ dị irè na-emetụta ihe mgbaàmà ndị dị otú ahụ dị ka delusions, mmegharị anya, ịmụ anya arọ nrọ, chere aghara, psychotic n'ahụhụ, omume aghara , na na. D. Kenye ndị a ọgwụ ọjọọ nwere ike na-nwetara dọkịta.

The kasị ewu ewu na antipsychotic ọgwụ eme "Chlorpromazine". Ntuziaka maka ojiji, price, reviews, analogs, megide-egosi na ọgwụ na-ọkọnọ n'okpuru.

Mejupụtara, nkọwa, ụdị

Olee ụdị bụ pụta ụwa ọgwụ "Chlorpromazine"? Ntuziaka, reviews na-akọ na a ọgwụ na-na-ere ụdị brownish-pink mkpụrụ ọgwụ, nakwa dị ka ihe ngwọta maka igba ogwu n'akwara na intramuscular ochichi. N'ọrụ umi pụtara data bụ chlorpromazine hydrochloride. Ọzọkwa, dabere na ntọhapụ n'ụdị ha nwere a dịgasị iche iche nke mgbakwunye.

pharmacological atụmatụ

Gịnị dị ịrịba ama iji ọgwụ "Chlorpromazine"? Ntuziaka maka ojiji, Ibọrọ na-egosi na nke a bụ ihe antipsychotic gị n'ụlọnga, nke site na ya pharmacological otu na-ezo aka neuroleptics. Ọ nwere a hypotensive, antiemetic na antihistamine mmetụta.

The n'ọrụ mgwa nke a ọgwụ bụ a emepụta nke phenothiazine. Tụkwasị na nke a Njirimara ifịk agwọ ọrịa nwere ogwuura, hypothermic-adịghị ike, antipsychotic, obodo iwe, vasodilating na moderately M-anticholinergic mmetụta.

Antipsychotic mmetụta nke ngwá ọrụ na-enweta site igbochi dopamine D 2 anabata na mesolimbic systems Mesocortical. N'ihi dị otú ahụ Njirimara nke ọgwụ bụ enwe ike iwepụ ịmụ anya arọ nrọ, delusions na ndị ọzọ na-arụpụta ihe mgbaàmà nke psychosis.

Ọ ga-kwuru nakwa na "Chlorpromazine", reviews nke nke na-depụtara n'okpuru ebe a, aka dị iche iche na iche nke psychomotor n'ahụhụ, ime ihe ike na-ebelata ịdị njọ nke psychotic egwu.

Ogwuura mmetụta nke ọgwụ na-enweta site igbochi adrenergic reticular ahịa ọgwụ na-emi odude ke brainstem.

Njirimara nke ọgwụ

Gịnị bụ Njirimara pụta ụwa na agwọ ọrịa "Chlorpromazine"? Nyocha kọrọ na a ọgwụ a nkụda mmụọ na oyi mpiaji ọrụ, eme ka ndị skeletal mọzụlụ, ebelata n'amaghi moto ọrụ, na-ebelata uche na endogenous na exogenous stimuli na a otu ebe uche. The ojiji nke nnukwu doses nke ọgwụ na-akpata oké iro ụra.

Mgbochi nke vagus akwara na eriri afọ tract na dopamine D2 anabata emi odude ke emetic akpalite na mpaghara na center enye antiemetic mmetụta nke ọgwụ ahụ. Ọ kwesịkwara kwuru na nke a owuwu nwere obere mmetụta M-cholinergic anabata. Ọzọkwa, ya akpọ mmetụta hụrụ maka Alfa-adrenergic anabata.

The edinam nke ọgwụ

ọgwụ ọjọọ, "Chlorpromazine" Olee otú ọ na-arụ ọrụ? Nyocha na-ekwu na ngwá ọrụ a na-enwe ike kpam kpam wepụ mmetụta na e mere site epinephrine. Ya hypothermic mmetụta n'ihi mgbochi nke dopamine anabata na-emi odude ke hypothalamus.

E lee ya anya ọgwụ lowers ọbara mgbali, obi ọnụego na-abawanye, nwere a na-adịghị ike antihistaminic mmetụta na owụt kataleptogennoe edinam, na-ebelata permeability nke capillary mgbidi.

N'ihi na intramuscular ochichi na agwọ ọrịa na-akpata ogwuura n'oge ¼ awa, na mgbe onu ochichi - mgbe 120 nkeji. Ndidi ndidi na ogwuura na hypotensive mmetụta amalite na banyere otu izu.

Mgbe ị na-enweta nke a ọgwụ n'ime ya antipsychotic Njirimara nwere mmetụta na 4th ma ọ bụ 7th ụbọchị. The ọgwụgwọ mmetụta nke ọgwụ dịruru banyere 2-6 ọnwa.

The pharmacokinetics nke ọgwụ

Ndi "Chlorpromazine" ṅụrụ? Nyocha akọ na ihe ọnụ chlorpromazine ngwa ngwa ma ọ bụghị kpamkpam etinye obi gị dum na digestive usoro. Ya elu ọbara kasịnụ enweta mgbe 4 h.

A ọgwụ dabara mbụ gabiga imeju. Ya mere ya ịta n'ime ọbara mgbe onu ochichi nnọọ obere karịa ịta mgbe intramuscular ochichi.

The ọgwụ na-metabolized na imeju na-adịghị ejekwa ozi na-arụsi ọrụ ike emepụta.

Chlorpromazine nwere nnukwu nkekọ na-plasma-edozi. Ọ na-ekesa na ahụ onye ọrịa, na-abami site BBB.

Ọkara ndụ-nke na-arụ ọrụ bekee nke ọgwụ bụ banyere 30 nkeji. N'ihi ya mkpochapu ya emepụta nwere ike ịbụ ogologo oge.

Egosipụta agwọ ọrịa na-ewere ya na mmamịrị na bile.

Drug "Chlorpromazine": egosi maka ojiji

Nyocha kọrọ na ọgwụ na ọtụtụ-eji psychiatric omume. Ọ na-kenyere na ọgwụgwọ nke n'ahụhụ na onye na isi mgbaka. Ọzọkwa, a ọgwụ na-eji na-adịghị ala ala psychosis, nnukwu nkwenkwe ụgha na-ekwu, hypomanic mkpali, ehighi ura, psychopathy, echiche ọrịa, nchegbu, egwu na inwe nchekasị.

Na mgbakwunye na ọnọdụ e depụtara na-egosi maka ojiji nke a ọgwụ bụ: persistent hiccups, mmanya psychosis, enweghịkwa nchịkwa vomiting na oké ọgbụgbọ. Ọ bụrụ na e mgbu ọgwụ enhances mmetụta nke analgesics.

Ọ kwesịkwara kwuru na n'aka E Kenyere atụle ọrịa nke na-ebu ụba muscular ụda, tetanus (dị ka Nchikota ọgwụ na njikọ na barbiturates) na mgbe dị iche iche na-enwe nsogbu ọrịa ụbụrụ mgbasa.

Ọ bụghị otú ahụ ogologo oge gara aga, a ọgwụ na-eji maka wuru hypothermia ekewet lytic mixtures. Na na-akụnwụ ahụ a ọgwụ na-kenyere ogwuura na izugbe ná Nkụnwụ potentiation.

Na dermatological omume "Chlorpromazine" (Ibọrọ nke ọrịa banyere ọgwụ ndị tumadi mma agwa) eji na itching dermatoses. Ke adianade do, ọ ga-eji na ọgwụgwọ nke nnukwu porphyria agwa.

contraindications

Mgbe ụfọdụ, adịghị kenyere antipsychotic "Chlorpromazine"? Nyocha nke dọkịta na-akọ na ngwá ọrụ a na-adịghị eji na comatose ekwu ọ bụla na isi iyi, nakwa dị ka na-arịa ọrịa oké mmegbu nke ụjọ usoro, oké ọrịa obi na ọrịa na vaskụla ekweghị ibe nọrọ na-arụsi ọrụ ike umi, a na-aga n'ihu ọrịa nke ụbụrụ na spinal systemic ọdịdị nke ụbụrụ, ọnyá ọnya nke eriri afọ tract na n'oge ara nri.

Na echiche nke elu n'ihe ize ndụ nke hepatotoxic Jeremaya mere, ọ pụtara ọgwụ na oké ịkpachara anya na aṅụrụma. Otu bụ eziokwu ara cancer, ọbara dyscrasias, hyperplasia nke prostate gland, glaucoma, mechiri emechi-ụdị, ọrịa Parkinson, àkwụkwụ, myxedema, vomiting, cachexia, Reye syndrome na ndị agadi.

Drug "Chlorpromazine": ntuziaka maka ojiji

Mbadamba ratings nke na-ọkọnọ dịrị gaba n'ime ebe, eji na psychiatric omume na-amalite kwa onunu ogwu hà 25-100 mg. A ego ekewa 1-4 doses. N'ime oge ahụ, dịkwuo dose ọ bụla ụbọchị anọ nke 25 ma ọ bụ 50 mg nweta chọrọ mmetụta.

Nchegbu preoperatively ifịk ọgwụ ọṅụṅụ maka 2-3 awa.

The kacha otu dose nke gị n'ụlọnga bụ 300 mg, na kwa ụbọchị - 1,5 g

Banyere ihe ngwọta, ọ na-ndinọ intravenously ma ọ bụ intramuscularly. Mbụ onunu ogwu nke a ọgwụ bụ 25-50 mg.

Tupu ochichi nke ọgwụ ọ jiriwo 2.5 ml nke sodium chloride ngwọta ma ọ bụ procaine. Ọgwụ eme miri intramuscular ogwu ogbugba.

The kacha otu dose nke gị n'ụlọnga bụ 150 mg na kwa ụbọchị - 1 g Ma igba ogwu n'akwara ochichi, ndị a ụkpụrụ-ederịta akwụkwọ ozi 100 na 250 mg.

ekwesighi mmetụta

Eme ihe ọ bụla mmetụta "Chlorpromazine" (mbadamba)? Nyocha kọrọ na mmalite nkebi nke ọgwụgwọ a ọgwụ nwere ike ime ka akọrọ ọnụ, paresis nke ulo, frigidity, mụbara iro ụra, afọ ntachi, nsogbu ihi ụra, dizziness, mkpọchị agụụ, tachycardia, kwuru ụdị orthostatic hypotension, urinary njigide, belata potency, nke ahu anataghi na ọdịda ọbara mgbali.

Ruo ogologo oge ọgwụ na a ọgwụ na-akpata muscle cramps n'olu ma ire, neuroleptic ịda mbà n'obi Akinetes-isiike onu, extrapyramidal ọrịa, amenorrhea, akathisia, na-egbu oge mmeghachi omume dị iche iche stimuli, hypercoagulability, vomiting, iche echiche mgbanwe, gbasara obi arrhythmia, pigmentation nke anụ, mgbochi nke ụmị ọkpụkpụ hematopoiesis , gynecomastia, cholestatic jaundice, galactorrhea, giperplolaktinemiyu, oliguria, afọ ọsịsa, na neuroleptic ajọ syndrome. Na igba ogwu n'akwara infusion phlebitis kpụrụ na intramuscular - infiltrates.

kpọmkwem na-atụ aro

Agwọ nke ngwá ọrụ a na-achọ ịkpachara anya akara nke ọbara mgbali, usu, ọrụ nke akụrụ na imeju.

A ọgwụ nwere ike ime ka photosensitivity, ya mere na oge nke ya mbanye na-atụ aro iji zere ikpughe.

Analogs na-eri

The price nke a ọgwụ na-adabere na ntọhapụ ụdị. Packaging nke 10 vials nwere ike zụrụ n'ihi na 60 rubles, mgbe a yiri ọnụ ọgụgụ nke mbadamba bụ banyere 150 rubles.

Site analogues nke a ọgwụ na-agụnye "Chlorpromazine hydrochloride" na "Tisercinum".

Nyocha

Dị ka ndị ọkachamara lere ya anya na ndị agwọ ọrịa nwere ike antipsychotic mmetụta, okodorode niile ihe ịrịba ama nke psychomotor n'ahụhụ. Otú ọ dị, ọ ga-ahụ kwuru na nke a pụtara na reviews bụ nke dị iche iche agwa.

Ụfọdụ ọrịa na-ekwu na a ọgwụ bụ irè ọrịa Alzheimer, isi mgbaka, psychosis, Akwụkwụ na-adọ, na a na-aka nchekasị na nrụgide. Ndị ọzọ nwere na-eji ọkụ kwere na-ewere ọgwụ na-akpalite mmepe nke akwụkwụ ọdịdọ, n'aka-shake, dị iche iche na àgwà ọrịa na oké ụra ala.

Na nke ọ bụla, nke a usọbọ kwesịrị na-eji dị ka bu n'obi na n'okpuru nlekọta nke ịga dọkịta.

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