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Ọgwụ "Sporagal": ntuziaka maka ojiji, analogs na reviews

Olee na-ọgwụ ọjọọ, "Sporagal"? Ntuziaka na ojiji nke ọgwụ ga-atụle n'ihu. Ị ga-amụtakwa ma e nwere analogues nke a nkwadebe, ole ọ na-efu, na-ekwu banyere ya ọrịa, ihe mere ọ na-ndinọ, na na. D.

Ụdị, mejupụtara, nkwakọ antifungal ọgwụ

Nkwadebe "Sporagal" dị na Capsule ụdị. Ya isi nọ n'ọrụ mgwa bụ itraconazole. Ọzọkwa na agwọ ọrịa mejupụtara polyethylene glycol 20000, sucrose, na hydroxypropyl acrylate copolymer.

Na-akwanyere ndị shei, ọ na-emi esịnede gelatin, titanium dioxide na indigotin.

Na a ngwugwu na-eresị na nkà mmụta ọgwụ "Sporagal"? Ntuziaka maka eji ngwá ọrụ a na-agbakwunyere na a kaadiboodu igbe. Ọ na-nwere a ike gelatin Capsule nke-acha anụnụ anụnụ (na blisters), nke nwere * Tụkwasị na nsogbu dị iche iche nke odo agba.

Pharmacodynamics agwọ ọrịa

Olee otú "Sporagal" mbadamba? Dị ka ntụziaka, ọgwụ bụ a emepụta nke triazole. Ọ nwere elu ọrụ megide dịkwa ka usoro ha.

The ọgwụ na-enyere nwayọọ na ndu njikọ nke ergosterol, na-enye ihe antifungal mmetụta.

Ọkachamara na-ekwu na itraconazole egbochi uto na mmeputakwa nke nnukwu ọnụ ọgụgụ ụdị dịkwa ka usoro ha.

The pharmacokinetics nke antifungal gị n'ụlọnga

Drug "Sporagal", nke analogues ga-kpọmkwem n'ihu, ngwa ngwa etinye obi gị dum n'ime n'ọbara. The kasị elu larịị nke itraconazole na ụmụ mmadụ na-hụrụ mgbe 3 awa. Ya bioavailability bụ 55% (kacha a hụrụ na n'ikuku capsules ozugbo oriri nke a abụba na elu-kalori oriri).

Itraconazole a na-ekesa dị iche iche akụkụ na anụ ahụ nke ahụ. Ya ọdịnaya na ọkpukpu, akụrụ, imeju, akpa ume, skeletal muscle, afo, splin na ugboro 3 elu karịa ọbara.

Agwọ ọrịa metabolized na imeju nyak a plurality nke emepụta. Otú ọ dị, naanị gidroksiitrakonazol nwere a akpọ antifungal mmetụta.

Odika 34% nke nọ n'ọrụ umi ẹkesiode ke mmamịrị, na banyere 54% site na eriri afọ.

Na ndị mmadụ na ihe isi imeju ọrụ na ọrịa akụrụ, na ọrịa na immunosuppression bioavailability nke ọgwụ nwere ike belata.

egosi capsules

Mere họpụta "Sporagal"? Ntụziaka na-ekwu na ọgwụ a na-zubere maka ọgwụgwọ nke fungal-efe efe, nke na-iwe na ọgwụ uche pathogens:

  • vulvovaginal candidiasis;
  • ophthalmological na dermatological ọrịa nke fungal si (e.g., fungal keratitis, ringworm, pityriasis versicolor);
  • onu candidiasis ;
  • onychomycosis, nke na-iwe na dermatophytes ma ọ bụ yeasts;
  • systemic mycoses tinyere cryptococcosis (ndị na-adịghị ike dịghịzi usoro n'oge ụjọ usoro cryptococcosis agwọ ọrịa ndinọ naanị na enweghị ọgwụgwọ mmetụta nke ndị ọzọ antifungal mmadụ), cryptococcal meningitis, systemic aspergillosis na candidiasis;
  • sporotrichosis, paracoccidioidomycosis, blastomycosis, histoplasmosis, na ndị ọzọ na obere systemic mycoses.

Contraindications ojiji nke capsules

Gịnị bụ contraindications na ojiji nke a ọgwụ ọjọọ, "Sporagal" (mbadamba)? Ntụziaka na-ekwu na ọgwụ ọ gaghị eji na:

  • Hypersensitivity ka isi na nke sekọndrị, mmiri nke ọgwụ
  • njikọ na ndị dị otú ahụ ọgwụ dị ka "Eletriptan" blockers HMG-CoA reductase inhibitors (e.g., "atorvastatin", "Lovastatin" "simvastatin"), ergot alkaloids, substrates CYP3A4 (atụ, "Cisapride", "bepridil," "pimozide" "Dofetilide", "Astemizole" "quinidine" "mizolastine"), "nisoldipine," "Midazolam", "triazolam".

Ọ kwesịkwara kwuru na ojiji nke a ọgwụ na-contraindicated n'ihi na ndị mmadụ na ventricular dysfunction na obi ọdịda, karịsịa congestive agwa.

Drug "Sporagal": ntuziaka maka ojiji

Dị ka ntụziaka, ọgwụ kwesịrị naanị iwere ọnụ. The capsules ga-iwesa ozugbo a nri (iji hụ na mma absorption), na dum, na-enweghị ịta.

The onunu ogwu nke a ọgwụ na-adabere na ụdị ẹdude ọrịa:

  • Dermatological na ophthalmologic lesion (e.g., pityriasis versicolor ma ọ bụ ringworm) - 200 mg otu ugboro n'ụbọchị ruo otu izu.
  • Keratinized ọnya nke anụ (aka na ụkwụ) - 200 mg ugboro abụọ n'ụbọchị nke a izu.
  • Vulvovaginal candidiasis - 200 mg ugboro abụọ n'ụbọchị ruo ụbọchị atọ.
  • Oral candidiasis - 100 mg otu ugboro n'ụbọchị izu abụọ. Na ọrịa na AIDS ma ọ bụ neutropenia, dose ụba 200 mg otu ugboro n'ụbọchị.
  • Fungal keratitis - 200 mg otu ugboro n'ụbọchị izu atọ.
  • Onychomycosis, nke e mere site dermatophytes ma ọ bụ yeasts, na-emeso site na nke ugboro ugboro ọmụmụ. Otu ọgwụ na-agụnye na-ewere abụọ capsules ugboro abụọ n'ụbọchị nke a izu. Maka ọgwụgwọ nke ntu ọnya na mkpịsị aka a rụrụ 2 ọmụmụ nke a ọgwụ, na na ụkwụ ya - 3 ọmụmụ. The ezumike n'etiti abụọ ga-3 izu. Mmetụta na-egosipụta mgbe N'ezie ẹkụre (na uto nke ntu efere).

Esi kpọpụ mmadụ nile nkwadebe "Sporagal" nke ntu na akpụkpọ a rụrụ maka ogologo oge karịa site na ọbara. Na nke a, ezigbo ọgwụgwọ mmetụta maka ọrịa na-enweta nanị mgbe izu atọ mgbe ẹkụre ọgwụ nke na-efe efe na ihe dị 9 ọnwa mgbe ọgwụgwọ nke onychomycosis.

Ụzọ nke Jiri nke capsules maka systemic ọnya

Dị ka systemic ọnya ebu ngwa? "Sporagal" ikpo na-eso Dosages:

  • Candidiasis - 100-200 mg ugboro kwa ụbọchị maka 5-30 izu.
  • Cryptococcosis enweghị meningitis - 200 mg kwa ụbọchị maka 3-12 ọnwa. Na abụọ dose meningitis.
  • Aspergillosis - 200 mg kwa ụbọchị maka 3-5 ọnwa.
  • Histoplasmosis - 200 mg ugboro abụọ n'ụbọchị ruo ọnwa asatọ.
  • Chromomycosis - 100-200 mg kwa ụbọchị n'ihi na ọnwa isii.
  • Sporotrichosis - 100 mg kwa ụbọchị ọnwa atọ.
  • Paracoccidioidomycosis - 100 mg kwa ụbọchị n'ihi na ọnwa isii. Maka AIDS ọrịa, na onunu ogwu nwere ike ụba.
  • Blastomycosis - 100-200 mg ugboro abụọ n'ụbọchị ruo ọnwa isii.

Mmetụta nke ọgwụ

È nwere mmetụta na ọrịa na-anata "Sporagal" ọgwụ ọjọọ? Nyocha ọkachamara kọrọ ndị na-esonụ kwuru:

  • neutropenia, thrombocytopenia, leukopenia;
  • akụkụ okuku ume na tract-efe efe (elu);
  • hypertriglyceridemia, hypokalemia, hypocalcemia;
  • isi ọwụwa, paresthesia, elu neuropathy, hypoesthesia, dizziness;
  • ọbara ọrịa, angioneurotic edema, anaphylactic na anaphylactoid nfụkasị Jeremaya;
  • bịara ikiri ọhụụ, diplopia, ikpe ọnwụ, tinnitus, bịara ikiri ọhụụ;
  • obi ọdịda, karịsịa congestive agwa;
  • dyspnea, rhinitis, Sinusitis, akpa ume edema;
  • vomiting, dyspepsia, hepatotoxic Jeremaya mere, abdominal mgbu, pancreatitis, ọgbụgbọ, dysgeusia, afọ ntachi, ịba ọcha n'anya, afọ ọsịsa, bloating, nwa oge nrigo nke imeju transaminases;
  • mgbu nkwonkwo na akwara;
  • ọkụ ọkụ, photosensitivity, leukocytoclastic vasculitis, alopecia, nsí epidermal necrolysis, pruritus, exfoliative dermatitis, ọkụ ọkụ, nnukwu generalized exanthematous pustulosis, erythema multiforme;
  • dysmenorrhea, urinary incontinence, erectile dysfunction, pollakiuria;
  • fever, edema.

kpọmkwem na-atụ aro

Ihe i kwesịrị ịma na-enwe ndidi, tupu ewere ọgwụ "Sporagal"? Ibọrọ kọrọ na ya nọ n'ọrụ umi nwere a na-adịghị mma inotropic mmetụta.

Mgbe na-ewere nke a ọgwụ nwere ike ịzụlite congestive obi ọdịda, na oké hepatotoxicity.

Mgbe belata acidity ọgwụ absorbability-adị njọ.

People n'out oge n'itinye antacids ga-nọgidere na-enwe n'etiti ha na ụzọ nke nkwadebe kọwara nkeji nke 2 awa.

Drug "Sporagal" na-atụ aro maka agadi ọrịa.

Ọ bụrụ na ị nwere mgbanwe nke elu neuropathy inweta ọgwụ iji kagbuo.

Ara na ime

N'oge ime, ọgwụ ike ga-ndinọ naanị na systemic mycoses, nke bụ a egwu egwu nne ndụ.

Ma ara, na oge a, "Sporagal" na-kwere, ma naanị n'okpuru ike na-egosi.

Drug "Sporagal": analogs na price

Na-esonụ ngwaọrụ bụ ihe ndị kasị mara analogues nke ọgwụ n'okpuru echiche, "Itrungar", "Sporaksol", "Orungal", "Eszol" na "Funit".

Ego ole ka a ọgwụ ọjọọ, "Sporagal"? The price nke a ọgwụ dịgasị n'etiti 1100-1200 rubles.

Nyocha nkwadebe

Dị ka nzaghachi nke ndị na-ada ọgwụ, ọ nwere ike kwuru na ọ bụ nnọọ irè-egosipụta onwe ya na dị iche iche nke fungal-efe efe. nwere ike kewapụrụ ọjọọ ozi bụ ndị na-ekwu na ngwá ọrụ a nwere a elu na-eri. Otú ọ dị, ndị ọkachamara na-ekwu na price nke a ọgwụ kpamkpam n'onye ezi omume site ya ọgwụgwọ nrụpụta.

Ma ihe ndị ụkọ ihe ụfọdụ nke a ọgwụ, ndị ọrịa na-arụtụ aka dịtụ ogologo oge ọgwụgwọ.

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