Ahụ ike, Preparations
"Ereksezil": ikom reviews, ntuziaka maka ojiji, a nkọwa nke analogs
A ọ na-ọgwụ ọjọọ bụ "Ereksezil"? Nyocha nke ikom banyere irè nke ego a ga-atụle mgbe e mesịrị na isiokwu. Ị ga-amụtakwa banyere ihe nwere ike dochie kwuru agwọ ọrịa n'ụdị nke ọ na-emepụta na ihe nwere pharmacodynamic Njirimara.
Mejupụtara nkọwa ọgwụ ụdị na Products
"Ereksezil" - mbadamba-acha anụnụ anụnụ na oval ekara, film-ntekwasa (film). Ha bụ isi n'ọrụ mmewere bụ sildenafil citrate. Ọzọkwa kwuru agwọ ọrịa mejupụtara ndị na-esonụ inyeaka Efrata: microcrystalline cellulose, croscarmellose sodium, calcium hydrogen phosphate na mg stearate.
Banyere-acha anụnụ anụnụ n'ọbọ, ọ bụ-acha anụnụ anụnụ Opadry II 85F20464 (i.e. polyvinyl mmanya, macrogol, titanium dioxide, talc, indigo carmine aluminum ghọọ).
The ire ọgwụ ọjọọ "Ereksezil" (Ibọrọ nke ndị ikom bụ karịa mma agwa) abịa na ọnya Ukwu, nke na-packaged ke Ukwu nke kaadiboodu.
Ụkpụrụ nke edinam nke ọgwụ
Erectile dysfunction - ọ bụ a nsogbu nke ọtụtụ oge a na ndị ikom. Ya mere, na-emepụta ọgwụ na ụlọ ọrụ ndị na-emepe emepe ọzọ na ndị ọzọ ọgwụ ọhụrụ maka ọgwụgwọ nke si ala. Otu n'ime ha bụ ụzọ nke "Ereksezil". Nyocha nke ndị ikom na-akọ na ọgwụ dị mma na ngwa ngwa na-eweghachi mkpọchị erectile ọrụ ma na-enye a nzaghachi mmekọahụ mmalite.
Irè nke a ọgwụ ruru ya mejupụtara. Sildenafil bụ n'ọrụ mgwa nke ọgwụ. Ọ bụ a nhọrọ ma nke nwere ike inhibitor nke cGMP-kpọmkwem PDE5, nke bụ maka na mmebi nke cGMP na cavernous ahu.
Sị na akụrụngwa ọ dịghị ihe kpọmkwem-atụrụ ndụ ihe na corpus cavernosum, ma enhances budata NO izuike utịp ke anụ ahụ.
N'oge mmekọahụ agụụ mmetụta obodo ntọhapụ nke nitric oxide eme sildenafil PDE5 mgbochi, na-amụba ọdịnaya nke cGMP na cavernous ahu. N'ihi ya, e ime ụba ọbara na-eji ire ụtọ muscle ntụrụndụ.
Ndị ọzọ na-ọgwụ
The ịrịba ama "Ereksezil" Erere maka ndị ikom? The n'ọrụ mgwa nke a ọgwụ bụ mgbe na-akwụsị akwụsị ischemic iche na agba dị ka acha anụnụ anụnụ na green. A mmetụta yiri jikọtara mgbochi nke ndị ọkachamara PDE6, nke na-na abuana ke nnyefe nke ìhè na visual akụkụ.
The kinetic Njirimara nke ọgwụ
Olee ihe nwere kinetic ọgwụ "Ereksezil", analogues nke nke na-depụtara n'okpuru ebe a? Dị ka ntụziaka, mgbe ochichi n'ime ya n'ọrụ mgwa na-etinye obi gị dum ngwa ngwa. The zuru bioavailability nke ọgwụ bụ banyere 41%.
Mgbe anata sildenafil ọnụ na a ọdụdụ nri ya absorption ọnụego na-ukwuu belata. Sị na umi, na ya isi metabolite 96% ibikwa na plasma-edozi.
Sildenafil na-metabolized n'okpuru nduzi imeju microsomal isozymes. Ya ọkara ndụ bụ banyere awa anọ.
egosi maka
Preparations maka potency dị nnọọ ewu ewu n'etiti ndị na-ata ahụhụ site na erectile dysfunction. "Ereksezil" na-aduak na-emeso a ọrịa ji enweghi ike nweta na iji nọgide na ihe erection nke amụ zuru ezu maka na-eju afọ-enwe mmekọahụ.
N'ihi ya, ọ bụ nchebe iji mara na Sildenafil egosipụta elu arụmọrụ naanị mgbe agụụ mmekọahụ na mmalite.
Bans ojiji nke
Mgbe ụfọdụ, i nwere ike iji ọgwụ ọjọọ eme ihe maka potency? Mbadamba "Ereksezil" contraindicated na-enweta na:
- imekotaotuugbo ojiji nke ọgwụ ọjọọ ndị ọzọ maka ọgwụgwọ nke erectile dysfunction (nrụpụta na nchekwa nke sildenafil dị otú ahụ ihe n'ịgwa na e mụọ);
- mgbe nile ma ọ bụ intermittent ojiji nke donators NO, organic nitrati ma ọ bụ nitrites n'ụdị ọ bụla (ebe sildenafil enhances antihypertensive mmetụta nke nitrati);
- dị ka a obere;
- concomitantly na ritonavir;
- elu uche nke onye ọrịa na sildenafil ma ọ bụ ndị ọzọ akụrụngwa nke ọgwụ.
Ọ kwesịkwara kwuru na kwuru n'aka na-aju ekenye nwanyi mmadụ.
Kpachara anya ngwa
Anya mbadamba "Ereksezil" ga-eji obi ọdịda, anatomical deformation nke amụ, ọrịa na predispose na mmepe nke priapism ọchịchọ ọbara ọgbụgba, ejighị n'aka rịaworo, exacerbation nke peptic ọnyá afọ nke digestive tract, ọrịa strok, butere n'aka retinitis pigmentosa, myocardial infarction, arrhythmias, egwu ndụ, hypotension, ọbara mgbali elu, ischemic optic neuropathy.
Mbadamba "Ereksezil": ntuziaka maka ojiji
Weere a ọgwụ kwesịrị naanị iwere n'ime. The na-atụ aro usoro onunu ogwu nke a ọgwụ maka ọtụtụ ndị toro eto bụ 50 mg 60 nkeji tupu mmekọahụ. Na echiche nke tolerability na nrụpụta ọrụ nke ọgwụ ọjọọ na dose nwere ike mụbara ruo 100 mg ma ọ bụ na-ebelata 25 mg.
Oke kwa onunu ogwu nke ọgwụ bụ 100 mg, na kacha na-atụ aro ojiji multiplicity - 1 oge kwa ụbọchị.
Ndị agadi dose ukpụhọde ọgwụ "Ereksezil" bụ chọrọ.
Na ọnụnọ nke gbasara akụrụ odida, agafeghị oke ma ọ bụ nwayọọ onunu ogwu ukpụhọde bụ chọrọ ma. Banyere oké gbasara akụrụ insufficiency, mgbe ahụ, na ala dose of sildenafil 25 mg.
Nyere na mkpochapu nke ọgwụ na-atụle isi na ndị na-imeju mmebi, ya ego a ga-ebelata ka 25 mg.
Mgbe imekotaotuugbo ochichi na ritonavir kacha otu dose of sildenafil ekwesịghị n'elu 25 mg, na ya multiplicity nke ngwa - 1 oge n'ime ụbọchị 2.
Na ihe yiri ngwa nke ọgwụ na inhibitors nke cytochrome CYP3A4 isoenzyme ya na-atụ aro amalite dose bụ 25 mg.
Iji belata ihe ize ndụ nke postural hypotension na ndị na-na-ewere Alfa-blockers, iji ọgwụ ọjọọ eme ga-atụle nanị mgbe mmalite nke hemodynamic stabilization. Ọzọkwa na nke a ga-atụle mkpa ime ka belata mbụ onunu ogwu nke sildenafil.
Ebibi site-agwa
Gịnị iwe nwere ike ime ka ọgwụ "Ereksezil", ego nke nke na-depụtara n'okpuru? Na ịdọkapụta ntụziaka nwere ndị na-esonụ na-akpata:
- gọzie gị mkpọchi, isi ọwụwa, arthralgia, na-ekpo ọkụ mgbukepụ, Sinusitis, dizziness, rhinitis, ehighi ura;
- pharyngitis, dyspepsia, myalgia, ọhụụ mgbanwe, ike ọgwụgwụ, na-eku ume nsogbu, afọ ọsịsa;
- ụba Akwara ụda, abdominal mgbu, conjunctivitis, ọgbụgbọ, akụkụ okuku ume na tract-efe efe;
- urinary tract ọrịa, flu syndrome, azụ mgbu, na mmepe nke na-efe efe ọrịa, priapism, vasodilation mgbaàmà, ọrịa nke prostate gland, anụ rashes.
Isi ihe ịrịba ama nke ovadozu
Mgbe na-ewere otu eji ọgwụ na a onunu ogwu nke 800 mg achọghị Jeremaya mere bụ tụnyere ndị mgbe na-anata agwọ ọrịa na ala doses, Otú ọ dị, ihe ndị ọzọ ọsọ.
The isi ihe nke a ọgwụ ovadozu agụnye ụba ogo mmetụta. Na omume dị otú ahụ symptomatic ọgwụ. Ọ kwesịkwara kwuru na dialysis anaghị mee ngwangwa ndị nwechapụ nke sildenafil. Nke a bụ n'ihi na eziokwu na-arụsi ọrụ ike umi "Ereksezila" ewee plasma-edozi na-anyụpụ site na akụrụ ya.
ọgwụ interactions
Dị ka ndị ọzọ ọgwụ ọjọọ eme ihe emekọ sildenafil? Dị ka ntụziaka nkwadebe "Cimetidine" ike dịkwuo ịta nke kwuru umi ke plasma site banyere 56%.
A otu ngwa "Ereksezila" ọnụ na erythromycin enwekwu AUC nke mbụ 182%.
Ke ukem ka n'ikuku nke saquinavir na sildenafil kacha ịta mụbara site 140%, a AUC na-amụba site 210%. N'ihi ya, chemical na ajụjụ na-enweghị mmetụta na kinetics nke saquinavir.
Siri ike otú ahụ inhibitors nke cytochrome CYP3A4, dị ka "Itraconazole" na "ketoconazole", na-eme mgbanwe ndị pụtara ìhè sildenafil pharmacokinetics.
A otu dose of antacid ahụ emetụtaghị bioavailability nke n'ụlọnga. Na nke a, sildenafil enhances hypotensive mmetụta nke nitrati. Na nke a, na ojiji nke a umi na Nchikota na nitrati na NO donators contraindicated.
Ụfọdụ mwute ndị na-na-enweta Alfa-blockers, concomitant ojiji nke sildenafil akpatakarị symptomatic hypotension.
Aṅụ na-ewere mbadamba antihypertensive ọgwụ adịghị akpata ọzọ mmetụta.
Olee ihe ndị ọzọ ọgwụ ọjọọ na mmekọrịta nwere "Ereksezil"? Mmanya mgbe na-ewere nke a na nkà mmụta ọgwụ na-machibidoro iwu. Ma ọ bụghị irè nke ọgwụ na-n'ụzọ belata.
Maka ozi ọzọ,
Tupu ịmalite na-ewere "Ereksezila" dị mkpa na-akpa àgwà a nyochaa nke CCC.
Weere a ọgwụ ghara ga-eji na ndị mmadụ n'ihi na onye mmekọahụ bụ ekwesighi.
-Nọgide kwuru mbadamba ọgwụ ndị na a ọchịchọ ọbara ọgbụgba.
Sildenafil enweghị mmetụta na a ikike mmadụ nwere iji ụgbọala ugbo ala na-arụ ọrụ ndị ọzọ usoro.
Analogs na ụlọ ọrụ na-akwụ ụgwọ
Site analogues ọgwụ "Ereksezil" na-agụnye ọgwụ ndị dị otú ahụ dị ka "Viagra", "Tornetis", "Viasan-LF", "Taksier", "Viatayl", "sildenafil", "Vigrande", "Silafil", "Vizarsin", " Ridzhamp "," Vildegra "," Revatsio "," ike "," Olmaks Strong "," Maksigra "na ndị ọzọ.
Ole a na-ewere a na nkà mmụta ọgwụ maka ọgwụgwọ nke ọrịa nke potency? The price nke a ọgwụ dị iche iche pharmacies nwere ike ịdị iche iche. Otú ọ dị, ná nkezi uru bụ mkpokọta 715 rubles (4 mbadamba 50 mg).
Drug "Ereksezil": ikom reviews
Gịnị ka ha na-asị ndị mmadụ nke ndị dị otú a ọgwụ dị ka "Ereksezil"? Kasị reviews nke atụle agwọ ọrịa bụ nanị mma. Men na-arụ ụka na ọ bụ a ukwuu irè ọgwụ, e mere ngwangwa mgbake nke isi erectile ọrụ, nakwa dị ka na-enye a eke omume mmekọahụ mmalite. Ọ bụ zuru ezu iji naanị otu mbadamba "Ereksezila" dị ka ike na mmekọahụ ozugbo kwuru ya irè edinam.
Ma ihe ndị na-adịghị mma na-akọ banyere nke a ọgwụ ọjọọ, ọtụtụ mgbe ha na-ezo aka n'eziokwu ahụ bụ na a ọgwụ nwere ike ime ka ọtụtụ mmetụta. Ke adianade do, ụfọdụ ọrịa na-enweghị afọ ojuju na elu na-eri ego, nyere na na a katọn ùkwù bụ nanị anọ stimulant mkpụrụ ọgwụ.
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