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Ọgwụ "Lamikon": ntụziaka, ngwa reviews, analogues, mejupụtara

Ego ole ka a ọgwụ dị ka "Lamikon"? The price nke a ọgwụ ga-ọkọnọ a n'isiokwu a. Ọzọkwa n'ebe ahụ ka ị ga-ahụ nkọwa zuru ezu ntuziaka maka ojiji nke ọgwụ, ya contraindications, analogs, na-egosi, oghom Jeremaya mere, ntọhapụ ụdị, Ọdịdị na na.

The mejupụtara, na udi ma na nkwakọ ọgwụ

Nweta atụle ọgwụ nwere ike ịbụ na ndị na-esonụ iche:

  • "Lamikon" aerosol. Ịgba nwere n'ọrụ umi dị ka terbinafine. Dị ka ndị ọzọ mmiri nke n'ụdị na-propylene glycol, macrogol cetostearyl ether 20, benzoic acid, disodium edetate, na mmiri ọgwụ Poloxamer 407. epicutaneous ọgwụ na-wepụtara na a kalama na a metering mgbapụta na 25 g.
  • Ude "Lamikon" (ude). Guide na-akọ na ndị nọ n'ọrụ mmewere nke a n'ụdị na-eje ozi terbinafine. Ọzọkwa Efrata nke a n'ụdị bụ: ịnweta mmanụ, sodium hydroxide, ọcha soft paraffin, cetostearyl mmanya na phenylethyl, macrogol cetostearyl ether 20, propylene glycol, poloxamer 407 na ọcha mmiri. Na ire nke manu-otite-abịa na akpa nke 15 g
  • "Lamikon" onu nkwadebe. Mbadamba, ntụziaka nke a na-nchọ na a igbe mere nke katọn, ịnwekwa dị otú ahụ na-arụsi ọrụ umi bụ terbinafine. N'ihe gbasara ndị ọzọ mmiri, ha na-agụnye: ọka starch, sodium starch glycolate, microcrystalline cellulose, colloidal anhydrous silica, hydroxypropylmethylcellulose na magnesium stearate. The mbadamba na-ẹdude ke sel nke ngwe nke 7 iberibe.

pharmacodynamics

Pharmacological otu atụle ọgwụ - antifungal. Dị ka ntụziaka, isi mgwa nke a gị n'ụlọnga bụ alilamin nke na-egosipụta na-arụsi ọrụ ọgwụgwọ mmetụta dị ukwuu nke dị iche iche dịkwa ka usoro ha pụta.

The fungicidal Njirimara nke terbinafine (nkịtị ịta) na-ekesa na dermatophyte dịkwa ka usoro ha, nakwa dị ka ụfọdụ ụdị nke dimorphic dịkwa ka usoro ha.

Dabere ụdị, megide yeasts a na nkà mmụta ọgwụ nwere ike igosipụta ma fungicidal na fungistatic ọrụ.

ụkpụrụ nke ime ihe

Olee otú ọgwụ "Lamikon"? Guide na-akọ na a gị n'ụlọnga kpọmkwem egbochi n'oge ogbo nke sterol biosynthesis na fungal cell membranes. The N'ihi nke ndị dị otú ahụ n'ebe na ihu ọma intracellular ìgwè squalene, na a enweghị ergosterol. Nke a na-eduga ná mbibi nke fungal mkpụrụ ndụ.

The usoro nke ihe nke ego na-ejikọrọ na usoro nke mgbochi nke enzyme squalene epoxidase ka, nke akọ na a cytochrome P-450.

Dị ka ọkachamara, ọgwụ ọjọọ, "Lamikon" enweghị mmetụta na mmetụta nke ndị ọzọ ọgwụ ọjọọ eme ihe, na mmiri ọgwụ metabolism.

Pharmacokinetics

Dị ka ọgwụ na-etinye obi gị dum, "Lamikon"? Guide na-ekwu na mgbe ndị obodo ma ọ bụ Nde ngwa absorption nke nọ n'ọrụ umi bụ ihe na-erughị 5% nke dose eji. Ya mere, ya systemic ikpughe bụ ala.

Mgbe ndinọ topically ọgwụ ozugbo amalite nwere mmetụta na bụ ukwuu irè maka a obere oge (ihe dị ka 8-13 ụbọchị).

Site n'idebe chọrọ ịta nke ọgwụ na stratum corneum nke epidermis, nke e nwetara n'oge ọgwụ, ndị fungicidal ihe nke agwọ ọrịa na-aga n'ihu n'ihi na otu onye izu mgbe ya kagbuo.

Mgbe e ji ọnụ na, "Lamikona" ifịk ifịk umi accumulates na anụ ahụ, mbọ na ntutu isi. Ịta nke ọgwụ na anụ ahụ kpamkpam na-enye ya fungicidal Njirimara.

Absorption nke mbadamba bụ 70%, na ha kpam kpam bioavailability - 50%.

The natara Nwa ke ichekwa 250 mg bụ ndị kasị elu ịta n'ime ọbara mgbe a ọkara awa. The irè ọkara ndụ oge banyere 30 awa.

The nri na ubé emetụta bioavailability nke ọgwụ. Na plasma protein ejikọ na-arụsi ọrụ ike umi nke 99,5%. Ọgwụ kama ngwa ngwa penetrates na dermis na accumulates na stratum corneum.

Nkewapụ iche "Lamikona" rụrụ site sebaceous glands. Ọzọkwa, ọ na-hụrụ na ntutu isi, akpụkpọ ntutu follicles. Ke akpa izu nke ọrịa, ọgwụ penetrates ntu efere.

Terbinafine na-metabolized ngwa ngwa na cytochrome P 450. Mgbe biotransformation ngwaahịa ewepụtara na-adịghị ejekwa metabolites site na akụrụ ya.

Mgbe ihe nhata na imeju na-na akụrụ nwechapụ nke terbinafine ọsọ slows budata, na-eme ya a elu ịta na plasma.

egosi

Malite mgbe ahụ inye obodo onunu ogwu forms "Lamikon" ọgwụ ọjọọ? Ude, ntuziaka maka ojiji nke a kọwara n'okpuru ebe a, nakwa dị ka ịgba nwere ndị na-esonụ na-egosi:

  • fungal anụ ọnya, nke e mere site na fungi nke genus Trichophyton, Microsporum na Epidermophyton (dermotofitiya ụkwụ, ukwu, toso, wdg);
  • multicolor (ma ọ bụ pityriasis) versicolor, nke malitere site na mmetụta nke Malassezia dịkwa ka usoro ha;
  • candidiasis nke anụ ahụ, nke triggered site dịkwa ka usoro ha nke genus Candida.

N'ihi nzube dị aṅaa na-eji onu forms "Lamikon" (mbadamba) nke ọgwụ? Guide na-akọ ndị na-esonụ na-egosi:

  • fungal-efe efe nke anụ ahụ, ebe ha njupụta, ịta ma ọ bụ okwu dị ka ha si na-emeso kpọmkwem onu uzo (naanị ekpebi dibịa);
  • mycosis isi na onychomycosis (ntu na-efe efe efere).

Ọ ga-kwuru na "Lamikon" mbadamba na-adịghị eji maka ọgwụgwọ nke acha (ma ọ bụ scaly) zoster.

contraindications

Olee ụdị contraindications kwesịrị maara nke tupu ị na-eji ọgwụ ọjọọ, "Lamikon"? Guide kwuru na naanị zuru ukpan nke ụdị nile nke ọgwụ a na-ewere hypersensitivity ya umi.

Ma ndị na-oge nke afọ ime, nwata na ara, ha na-ikwu contraindications.

Ude "Lamikon": ntuziaka maka ojiji

Ndị dị otú ahụ iche nke ọgwụ, dị ka a ịgba, na manu-otite, na-atụ aro ha mpụga ngwa. Tupu iji ha maka ọgwụgwọ nke fungal ọrịa, ị ga akpa ọcha ma na-emetụta akụkụ akpụkpọ.

Dabere na ogo nke ọrịa na ụdị nje ọgwụ "Lamikon" (ude) etinyere ugboro abụọ n'ụbọchị. Aerosol na-eji otu ugboro.

The ude ga-na etinyere ọ bụghị naanị ka otụk akpụkpọ ero, kamakwa n'akụkụ ebe. Iji mepụta a usoro ọ bụ na-achọsi ike ka mkpa oyi akwa nwayọọ nwayọọ rubbing ude mkpuchite.

Ọ bụrụ na ndị na-efe efe na ọrịa na-esonyere metụ akwa ọkụ ọkụ (e.g., n'okpuru ara, ukwu, ike ma ọ bụ n'etiti mkpịsị aka), na-emeso ebe kwesịrị ikpuchi fere fere (chi).

The ojiji nke aerosol

Olee otú m ga-eji ịgba "Lamikon"? Nyocha ọkachamara na-akọ na ọ na-eji n'ókè zuru ezu na moisten site spraying na ebe-eju na fungi, nakwa dị ka ike ikpa n'akụkụ ya.

Na oge nke ọgwụ na-adabere na obodo media ọrịa ogo (ruo izu abụọ).

Relief onye ọrịa kwuru a ụbọchị ole na ole. N'ihi na ihe irè ọgwụgwọ a choro iji rube isi ike ntuziaka ghara uche ọzọ na ngwa ma ghara ịkwụsị omume nká. Ma ọ bụghị ya, e nwere a elu n'ihe ize ndụ nke nlọghachi azụ.

Olee na-mbadamba?

Pharmacological ìgwè nwere ndị ọgwụ tupu anyị, gosiri na ntuziaka. Ọ na-agwa banyere esi mee ka na ngwá ọrụ.

Dị ka a na-achị, "Lamikon" mkpụrụ ọgwụ kenyere ụmụ si 6 afọ, nakwa dị ka okenye ọrịa. Ịnata onu nkwadebe na-aga n'ihu ruo mgbe zuru ezu ofufe nke niile ihe mgbaàmà nke a fungal ọrịa (dabere na ọdịdị na ogo).

The n'efu nke agwọ ọrịa onunu ogwu n'ihi na ndị okenye bụ 250 mg, na n'ihi na ụmụ-erikpu 20-40 n'arọ - 125 mg. Na a nnukwu ibu nke nwa dị ka ọgwụ 250 mg nke ọgwụ.

Na oge nke ọgwụ na trichophytosis na akpụkpọ candidosis bụ 2-4 izu, na na Tinea pedis - 2-6 izu.

Fungal ọrịa isi na ahụkarị na ụmụ. Dị ka a na-achị, ha na-amenable ọgwụgwọ ma ọ bụrụ na ọgwụ na-eji na Dosages na-atụ aro site dọkịta otu ọnwa.

Onychomycosis ọgwụgwọ na-ewe izu 6 maka mbọ aka na 12 - n'ihi na mkpịsị ụkwụ ntu. N'okpuru belata uto nke ntu efere ọgwụ nwere ike ruo ogologo oge.

oghom Jeremaya mere

Obodo ọgwụ "Lamikon", analogues nke nke na-depụtara n'okpuru ebe a, nwere ike ime ka mgbaàmà ndị dị otú ahụ dị ka akpụkpọ ekpepụsị, ọkụ, itching, ihe mgbu, iyatesịt, mkpọchị pigmentation, erythema na jikọrọ ọnụ guzobere. Ha nwekwara ike na-enweta nfụkasị Jeremaya.

Mgbe anata mbadamba, na-esonụ ekwesighi mmetụta:

  • neutropenia, agranulocytosis, Lyell syndrome, pancytopenia, Stevens-Johnson syndrome;
  • thrombocytopenia, anaphylactoid Jeremaya mere, uto n'ọgba aghara, ihe mgbaàmà nke lupus, isi ọwụwa;
  • photosensitivity, paresthesia, hypoesthesia, neuralgia;
  • dizziness, mmetụta nke ozuzù ke afo, afọ ọsịsa, na ọnwụ nke agụụ;
  • exacerbation nke psoriasis, ọgbụgbọ, psoriasiform rashes, abdominal mgbu, myalgia;
  • urticaria, arthralgia, ọkụ ọkụ, generalized pustulosis, ntutu isi ọnwụ, na-abawanye nke imeju enzymes;
  • ike ọgwụgwụ, hepatobiliary dysfunction, jaundice, ịba ọcha n'anya.

Analogs na-eri nke ọgwụ

Ego ole ka a ọgwụ ọjọọ, "Lamikon"? The price nke a ọgwụ na-adabere na ya udi. Ude na ịgba nwere ike zụrụ maka 180-220 rubles, na mbadamba - maka 370-400 rubles.

Ma ogbo, n'etiti ihe dị irè ị pụrụ igbunye dị otú ahụ ego dị ka "Amorolak" salicylic acid. "Mikoseptin", "Nitrofungin", "Mikolak", "Exoderil".

Nyocha nke agwọ ọrịa

Nzaghachi si ndị na-eji ọgwụ ọjọọ, "Lamikon" bụ oké mma. Ọrịa na-akọ na ndị ọgwụgwọ nrụpụta ọrụ nke a ọgwụ e hụrụ maka ụbọchị ole na ole mgbe ya nọ iji. A, a fungal ọrịa na kpamkpam site na njedebe nke N'ezie nke ọgwụ.

Na oké ikpe, ndị dọkịta nwere ike ikwu na a jikọrọ onunu ogwu ụdị (e.g., mbadamba na manu-otite, ịgba na mbadamba).

Na mgbakwunye na mma ozi banyere "Lamikon" nkwadebe zukoro na-adịghị mma nzaghachi. Ha na-emekarị jikọrọ ya adịghị irè ya. Otú ọ dị, ndị ọkachamara na-ekwu na nke a bụ omume na naanị na ọgwụgwọ nke na-abụghị chebaara agwọ ọrịa dịkwa ka usoro ha ma ọ bụ mebie ihe. Ya mere, tupu n'itinye manu-otite, mbadamba ma ọ bụ ịgba na-atụ aro ka ha hụ dọkịta na guzosie causative gị n'ụlọnga nke fungal ọrịa.

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