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"Tolperisone" n'aka. Ntuziaka maka ojiji

Mbadamba "Tolperisone" na-agụnye a ìgwè nke ọgwụ ọjọọ, muscle relaxants. The agwọ ọrịa nwere a Central mmetụta. The ọgwụ nwere a akpụkpọ ahụ kwụsie ike ọrụ, akwara-akwadoghị akwado slows ịgbachi motoneurons na isi afferent emep uta eri. Nke a na-akpalite igbochi nke poly- na monosynaptic spinal-aghọ nkọ. The ọgwụ na-egbochi ahụ conduction nke excitation na ụbụrụ azuokokoosisi reticulospinal ụzọ. N'agbanyeghị nke mmetụta nke Central ụjọ usoro pụtara amụba elu ọbara. Mmepe nke a pụrụ isi kwuo ya nwere ike ịbụ n'ihi na mmetụta nke antiadrenergicheskim na antispasmodic ọgwụ. N'itinye ọgwụ ọnụ ọ na-ọma etinye obi gị dum na obere eriri afọ. Mgbe ọkara awa, otu awa kacha hụrụ kacha ịta nke ọgwụ na plasma. N'ihi persistemnogo owụt metabolism agwọ ọrịa bioavailability nke 20%. Disintegration nke ọgwụ pụtara na akụrụ na imeju. N'ụdị metabolites ka 99% anyụpụ na mmamịrị.

"Tolperisone" na nkà mmụta ọgwụ. Ntuziaka maka ojiji. na-agba akaebe

Kenye ngwaahịa na elu (pathologically) ụda ma spasm na striated muscle metụtara na akwara ozi organic daa ọrịa na ọnya nke pyramidal tract, ọrịa strok, multiple sclerosis, encephalomyelitis, gụnyere myelopathy. The agwọ ọrịa "Tolperisone" ntụziaka ntuziaka na-atụ aro ka reductive ọgwụgwọ mgbe arụmọrụ ke traumatology na orthopedics. Site na-egosi na-agụnye ụda ma muscle spasm, muscular contracture, nsogbu ọrịa na nweekwa usoro. Karịsịa, ọgwụ dị irè na lumbar na cervical mgbu syndrome, ogbu na nkwonkwo na nnukwu nkwonkwo, spondyloarthrosis, spondylosis. Na Nchikota na ndị ọzọ n'aka nkwadebe "Tolperisone 'na-atụ aro ntuziaka maka ojiji na ọgwụgwọ nke occlusive vaskụla ọrịa ụdị. Ndị a na-egosi gụnyere Raynaud ọrịa, thromboangiitis, ọrịa angiopathy, atherosclerosis. N'aka họpụtara ọrịa kpasue-enwe nsogbu innervation nke arịa: angioneurotic intermittent disbazii, akrozianoz.

"Tolperisone" ọgwụ. Ntuziaka maka ojiji

The ọgwụ na-iwere na mbụ dose of 50 mg bụghị karịa ugboro atọ n'ụbọchị. Nke nta nke nta na-amụba ichekwa rụrụ ọgwụ 150 mg 2-3 p. / Day. Na oge na-ekpebisi ike n'otu n'otu dabere na ọdịdị na ogo nke ọrịa ala nke onye ọrịa.

contraindications

Mbadamba "tolperisone" (Ibọrọ ndị ọkachamara na-akwado ya) na-adịghị kenyere ụmụ ọhụrụ n'okpuru afọ 18 afọ, ekweghị ibe nọrọ nke mmiri. Contraindications gụnyere ime na lactation. N'ihi ọnụnọ nke lactose na ọgwụ na-atụ aro ọgwụ ekweghị ibe nọrọ ma ọ bụ erughi nke umi.

"Tolperisone" n'aka. Ntuziaka maka ojiji. oghom Jeremaya mere

The na nkà mmụta ọgwụ na-akpalite isi ọwụwa, muscle adịghị ike, ọgbụgbọ, gastralgia (na-agba na ala onunu ogwu). Na ndabere nke ọgwụgwọ na-egosi hypotension, anabata mere site ekweghị ibe nọrọ.

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